NCLEX Drugs Immunity and Chemotherapy

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Natural Immunity

  • Present at birth
  • Protection provided by physical barriers:
  • Skin, mucus membranes
  • Phagocytic cells
  • NK cells

Specific Acquired Immunity

Production of antibodies against antigens

Active:

  • Having the infection or a vaccine / toxoid
  • Takes weeks to months to take effect

Passive:

  • Administration of preformed antibodies (immunoglobulins)

Major Cells of the Immune System

  • B cells — Produce antibodies
  • Macrophages & Dendritic Cells
  • –Phagocytosis
  • Helper T cells (CD4)
  • –Activate B cells
  • –Responsible for delayed hypersensitivity reaction
  • Cytotoxic T cells (CD8)
  • –Directly destroy target cells

 

Important: You can find the latest list of childhood vaccines (ages, side effects etc. from the cdc). Here is the link.

http://www.cdc.gov/vaccines/schedules/hcp/child-adolescent.html

 

MMR Vaccine

Therapeutic Uses:

  • Measles, Mumps, Rubella

Adverse Effects:

  • Local reactions (rash, fever, swollen glands)
  • Anaphylaxis

Contraindications/Precautions:

  • Allergies to eggs, gelatin, and neomycin
  • Hx of thrombocytopenia
  • Immunocompromised individuals
  • Recently received blood products or immunoglobulins

 

DTaP Vaccine

Therapeutic Uses:

  • Diphtheria, Tetanus, Pertussis

Adverse Effects:

  • Encephalopathy (fever, persistent crying)
  • Seizures
  • Local reaction at injection site

Contraindications/Precautions:

  • Severe febrile illness
  • Hx of anaphylaxis
  • Hx of encephalopathy 7 days after DTaP vaccination
  • Occurrence of seizures with 3 days of vaccination
  • Inconsolable crying (>3 hrs) within 48 hrs of vaccination

 

Hepatitis Vaccine

Therapeutic Uses:

  • Hepatitis A & B viruses

Adverse Effects:

  • Local reaction
  • Anaphylaxis

Contraindications/Precautions:

  • Hx of anaphylaxis
  • Allergy to Baker’s yeast

 

Varicella Virus Vaccine

Therapeutic Uses:

  • Varicella zoster virus (chickenpox)

Adverse Effects:

  • Varicella-like rash

Contraindications/Precautions:

  • Pregnancy
  • Cancer
  • Hx of allergy to neomycin or gelatin
  • Immunocompromised patients

Education:

  • Slight risk of virus being transmitted. If child develops rash after vaccination they should be presumed to be infected and appropriate precautions taken.

 

Inactivated Polio Vaccine

Therapeutic Uses:

  • Immune response to poliovirus

Adverse Effects:

  • Vaccine-related paralytic poliomyelitis
  • Local reaction

Contraindications/Precautions:

  • None

 

Influenza Vaccine

Therapeutic Uses:

  • Immunity to influenza strains in the vaccine

Adverse Effects:

  • Guillain-Barré syndrome (ascending paralysis, weakness of BLE, dyspnea)
  • Local reaction
  • Fever

Contraindications/Precautions:

  • Acute febrile illness
  • Hypersensitivity to eggs

 

Immune Globulin

Expected Action:                  Proto: Gamma globulin (IgG)

  • Passive immunity

Therapeutic Uses:

  • Immunodeficiency syndrome
  • Bone marrow transplantation
  • Measles, rubella, varicella exposure •           Chronic lymphocytic leukemia
  • Hep A, Hep B exposure

Adverse Effects:

  • Local reaction / hypersensitivity

Contraindications/Precautions:

Interactions:

  • Live viruses can lead to disease – avoid live viruses for 3 months following IgG

Education:

  • Administer in deep muscle / Date of exposure must be known (6 days measles, 7 days Hep B, 14 days Hep B)

 

Immunostimulants

Expected Action:                  Proto: Interferon Alfa, Aldesleukin, Interleukin 2

  • Enhance immune response / reduce proliferation of cancer cells

Therapeutic Uses:

  • Leukemia / melanoma / Kaposi’s sarcoma

Adverse Effects:

  • Flu-like symptoms / Marrow suppression, alopecia, cardiotoxicity, neurotoxicity
  • Hypotension

Contraindications/Precautions:

  • Hypersensitivity / pregnancy and lactation (C)

Interactions:

  • Theophylline (toxicity)
  • Zidovudine or retrovir ( neutropenia)
  • Antihypertensives ( hypotensive effect)

Education:

  • Refrigerate / Do not shake vial

 

Immunosuppressants

(General)

  • Act on helper T lymphocytes to suppress proliferation of B cells and cytotoxic T cells
  • For treatment of autoimmune disorders and to prevent organ rejection
  • –Rheumatoid arthritis
  • –Early type 1 diabetes
  • –Lupus
  • –Myasthenia gravis

Adverse Effects

  • Teratogenesis
  • increased risk of infection

Medications:

  • Cyclosporine (Gengraf, Neoral)
  • Tacrolimus
  • Glucocorticoids (prednisone)
  • Methotrexate
  • Cytotoxics (azathioprine)

 

Cyclosporine

Adverse Effects: Hepatotoxicity Nephrotoxicity (BUN, Creatinine, I&O)

Contraindications/Precautions:  Pregnancy / Recent live virus vaccination / Recent contact ĉ chickenpox or herpes

Interactions:

  • Phenytoin, phenobarbital, rifampin, carbamazepine, TMP-SMZ ([cycl] ò)
  • Ketoconazole, erythromycin, amphotericin ([cycl] ñ ð toxicity)
  • Amphotericin, aminoglycosides, NSAIDs (all nephrotoxic ð ñ renal damage)

Grapefruit juice (ñ [cycl] by 50%)

Nursing

  • Mix oral dose ĉ milk or OJ to ñ palatability
  • Admin initial dose over 2-6 hours

Monitor for hypersensitivity, stay ĉ pt. for 30 mins

 

Glucocorticoids

Adverse Effects:

  • Osteoporosis (use Ca2+& vitamin D supplements
  • Renal insufficiency (stop drugs immediately)

Fluid retention

Contraindications/Precautions:

Systemic fungal infections

Recurring live virus vaccines

Interactions:

  • K+-depleting diuretics (ñ hypokalemia)
  • NSAIDs (ñ GI ulceration)

Glucocorticoids (Promote hyperglycemia)

 

Proto: Prednisone, prednisolone

 

Azathioprine

Adverse Effects:

  • Bone marrow depression à neutropenia & thrombocytopenia

Contraindications/Precautions:

  • None listed in ATI

Interactions:

  • Allopurinol (delays inactivation of azathioprine)

 

Antihistamines

(General)

  • Action is on H1 receptors which blocks histamine release

Medications

  • 1st Generation:
  • Diphenhydramine (Benadryl)
  • Promethazine (Phenergan)
  • Dimenhydrinate (Dramamine)

 

2nd Generation:

  • Loratadine (Claritin)
  • Cetirizine (Zyrtec)
  • Fexofenadine (Allegra)
  • Desloratadine (Clarinex)

 

Therapeutic Uses:

  • Mild allergic reactions
  • Anaphylaxis
  • Motion sickness
  • Insomnia

 

Antihistamines

(1st Generation)

 

Expected Action:      Proto: Diphenhydramine, promethazine, dimenhydrinate

  • Block H1 receptors – prevent histamine release into small blood vessels & nerves

 

Therapeutic Uses:

  • Mild allergic reactions
  • Motion sickness
  • Anaphylaxis
  • Insomnia

Adverse Effects:

  • Sedation
  • GI discomfort
  • Anticholinergic effects (dry mouth, constipation)
  • Acute toxicity (flushed face, fever, tachycardia), children can have hallucinations, incoordination and seizures –> to treat –> Induce vomiting and give activated charcoal.

 

Contraindications/Precautions:

  • 3rd trimester, lactation, newborns / use cautiously in kids and elderly
  • Caution ĉ asthma, urinary retention, open angle glaucoma, & hypertension.

 

Interactions:

CNS depressants

  • EtOH
  • Benzodiazepines
  • Opioids
  • Barbiturates

 

Chemotherapy Agents

(Medications)

  • Nitrogen mustards —> cyclophosphamide
  • Platinum compounds —> cisplatin
  • Folic acid analog —> methotrexate
  • Pyrimidine analog —> cytarabine
  • Purine analogs —> mercaptopurine
  • Antitumor antibiotics —> doxorubicin
  • Mitotic inhibitors —> vincristine, paclitaxel
  • Topoisomerase inhibitors —> topotecan, irinotecan
  • Breast cancer —> tamoxifen (antiestrogen)
  • Prostate cancer —> leuprolide
  • Progestins —> megestrol acetate

Cytotoxic medications

  • Asparaginase
  • Hydroxyurea
  • Procarbazine

 

Chemotherapy Agents

(Side Effects)

  • Bone marrow suppression –tx — Avoid crowds, check for bleeding gums
  • GI discomfort –tx — Give antiemetic (ondansetron) with dexamethasone, metoclopramide or granisetron at outset
  • Alopecia –tx —   Occur 7-10 days after, persist max of 2 months’ after
  • Mucositis –tx — Frequent oral care, soft toothbrush, EtOH mouthwash
  • Reproductive toxicity –tx — Sperm banking, Avoid gravid on meds.
  • Hyperuricemia or inc uric acid –tx —   inc fluids, I&O, Give allopurinol if inc uric acid
  • Extravasation of vesicants such as carmustine, dactinomycin, daunorubicin, and vincristine

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